Average Dose: .25mg - 1mg per day
Half Life: 5 - 7 days
Water Retention: none
Aromatization: no
DHT Conversion: no
Anastrozole is not a steroid. It is a tablet form anti-aromitase
that is used by many body builders to help prevent bloating (edema) and
Gynecomastia (bitch tit) associated with the use of testosterone and
androgens. It can be used in place of Nolvadex,Clomid, etc.
Bodybuilders are using around .25mg to 1mg per day or .5mg to 1mg every
other day and are having good success with it.
The FDA approved uses are for the treatment of breast cancer in
post-menopausal women with disease progression following tamoxifen
therapy. Hypersensitivity to anastrozole are reasons not to use this
drug. If you have these problems please inform your doctor. Common side
effects are: shortness of breath, dizziness, diarrhea, vomiting,
headache, hat flashes, weakness, cough, dry mouth, skin rash, sweating,
abdominal pain and bone pain. Some less common symptoms are vaginal
bleeding, weight gain, tiredness, chills, fever, breast pain, and
itching. In case of an overdose, it is recommended to contact your
poison control center, trade name: Anastrozole ) is a drug indicated in
the treatment of breast cancer in post-menopausal women. It is used
both in adjuvant therapy (i.e. following surgery) and in metastatic
breast cancer. It has the effect of decreasing the amount of estrogen
that the body makes.
Anastrozole (Anastrozole)Anastrozole belongs in the class of drugs
known as aromatase inhibitors. It inhibits the enzyme aromatase, which
is responsible for converting androgens (produced by women in the
adrenal glands) to estrogen.
The ATAC (Anastrozole, Tamoxplex, Alone or in Combination) trial
represents a long-term follow-up study of 9366 women with localized
breast cancer who received either anastrozole, tamoxifen, or both.
After more than 5 years the group that received anastrozole had
significantly better clinical results than the tamoxifen group. The
trial suggested that anastrozole is the preferred medical therapy for
postmenopausal women with localized breast cancer that is estrogen
receptor positive.
Usage for men
While officially indicated for women, this drug has proven effective in
the off-label use of reducing estrogen (in particular and more
importantly, estradiol) in men. Excess estradiol in men can cause
benign prostatic hyperplasia, gynecomastia, and symptoms of
hypogonadism. Some athletes and body builders will also use Arimidex as
a part of their steroid cycle to reduce and prevent symptoms of excess
estrogen; in particular, gynecomastia and water retention.
Study data currently suggests that dosages of 0.5mg to 1mg of Anastrozole
a day reduce serum estradiol by about 50% in men, which differs from
the typical reduction in postmenopausal women. However, the reduction
may be different for men with grossly elevated estradiol (clinical data
is currently lacking).